GSK199
Product Specifications
CAS Number
1549811-53-1
SKU
C12959-5mg
Target
PAD
Applications
Metabolism
Molecular Formula
C24H28N6O2.ClH
Additionnal Information
GSK199 is a reversible, specific inhibitor of peptidyl arginine deiminase 4 (PAD4), with an IC50 of 200 nM without calcium. It is involved in histone citrullination and neutrophil extracellular trap formation, making it useful for studying autoimmune, cardiovascular, and oncological diseases.
Available Sizes
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