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PF-4989216

Product Specifications

CAS Number

1276553-09-3

SKU

C12863-5mg

Target

PI3K

Applications

PI3K/Akt/mTOR

Smiles

C1COCCN1C2=C (C (=C (S2) C3=NC=NN3) C4=C (C=C (C=C4) C#N) F) C#N

Molecular Formula

C18H13FN6OS

Additionnal Information

PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.

Storage Conditions

2 years -80 in solvent

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