EPZ004777
Product Specifications
CAS Number
1338466-77-5
SKU
C12626-5mg
Target
Histone Methyltransferase
Applications
Epigenetics
Smiles
CC (C) N (CCCNC (=O) NC1=CC=C (C=C1) C (C) (C) C) CC2C (C (C (O2) N3C=CC4=C (N=CN=C43) N) O) O
Molecular Formula
C28H41N7O4
Additionnal Information
EPZ004777 is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM in a cell-free assay and demonstrates >1,200-fold selectivity for DOT1L over all other tested PMTs. EPZ004777 induces apoptosis.
Storage Conditions
2 years -80 in solvent
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
![Rat Monoclonal Corin Antibody (MM0199-9H21) [Alexa Fluor 700]](https://cdn.genprice.uk/genprice/uk/genprice4.webp)
NBP2-12205AF700 0.1 mL
Rat Monoclonal Corin Antibody (MM0199-9H21) [Alexa Fluor 700]
Sign In for Pricing
View Details 
FY-AB48735-01 1 mL
Anti-Chromatin Assembly Factor 1, Subunit B (CHAF1B)
Sign In for Pricing
View Details FY-AB48735-02 100 µL
Anti-Chromatin Assembly Factor 1, Subunit B (CHAF1B)
Sign In for Pricing
View Details FY-AB48735-03 200 µL
Anti-Chromatin Assembly Factor 1, Subunit B (CHAF1B)
Sign In for Pricing
View Details