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TEPP-46 (ML265)

Product Specifications

CAS Number

1221186-53-3

Synonyms

CID-44246499, NCGC00186528

SKU

C12586-5mg

Target

PKM

Applications

Metabolism

Smiles

CN1C2=C (C3=C1C (=O) N (N=C3) CC4=CC (=CC=C4) N) SC (=C2) S (=O) C

Molecular Formula

C17H16N4O2S2

Additionnal Information

TEPP-46 (ML265, CID-44246499, NCGC00186528) is a potent activator of PKM2 in both biochemical (AC50 = 92 nM) and cell-based assays with high selectivity over PKM1, PKR and PKL.

Storage Conditions

2 years -80 in solvent

Available Sizes

Frequently Asked Questions

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