Selexipag

Product Specifications

CAS Number

475086-01-2

Synonyms

NS-304, ACT-293987

SKU

C09559-5mg

Target

Prostaglandin Receptor

Applications

GPCR & G Protein

Smiles

CC (C) N (CCCCOCC (=O) NS (=O) (=O) C) C1=CN=C (C (=N1) C2=CC=CC=C2) C3=CC=CC=C3

Molecular Formula

C26H32N4O4S

Additionnal Information

Selexipag (NS-304, ACT-293987) is an orally active, first-in-class, selective prostacyclin IP receptor agonist with Ki value of 260 nM for human IP, whereas Ki values > 10,000 nM are measured at the other human G-protein-coupled prostanoid receptors (EP1-4, DP, FP and TP) .