What is the catalog number for Bemcentinib (R428)?

The catalog number for Bemcentinib (R428) is C08899.

What sizes are available for Bemcentinib (R428)?

Bemcentinib (R428) is available in the following size(s): 1 mg, 5 mg, 50 mg, 200 mg, 1 g.

How many pack sizes does Bemcentinib (R428) come in?

Bemcentinib (R428) is available in 5 different pack sizes.

Is Bemcentinib (R428) in stock?

Bemcentinib (R428) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Bemcentinib (R428)?

Bemcentinib (R428) is requires dry ice shipping.

Bemcentinib (R428)

Product Specifications

CAS Number

1037624-75-1

Synonyms

BGB324

SKU

C08899-1mg

Target

Axl

Applications

Protein Tyrosine Kinase

Smiles

C1CCN (C1) C2CCC3=C (CC2) C=C (C=C3) NC4=NN (C (=N4) N) C5=NN=C6C (=C5) CCCC7=CC=CC=C76

Molecular Formula

C30H34N8

Additionnal Information

Bemcentinib (R428, BGB324) is an inhibitor of Axl with IC50 of 14 nM, >100-fold selective for Axl versus Abl. Selectivty for Axl is also greater than Mer and Tyro3 (50-to-100- fold more selective) and InsR, EGFR, HER2, and PDGFRβ (100- fold more selective) .