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RO4929097

Product Specifications

CAS Number

847925-91-1

Synonyms

RG-4733

SKU

C07902-5mg

Target

Beta Amyloid

Applications

Neuronal Signaling

Smiles

CC (C) (C (=O) NCC (C (F) (F) F) (F) F) C (=O) NC1C2=CC=CC=C2C3=CC=CC=C3NC1=O

Molecular Formula

C22H20F5N3O3

Additionnal Information

RO4929097 (RG-4733) is a γ secretase inhibitor with IC50 of 4 nM in a cell-free assay, inhibiting cellular processing of Aβ40 and Notch with EC50 of 14 nM and 5 nM, respectively. Phase 2.

Storage Conditions

2 years -80 in solvent

Available Sizes

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