What is the catalog number for BI-671800?

The catalog number for BI-671800 is C07211.

What sizes are available for BI-671800?

BI-671800 is available in the following size(s): 5 mg, 25 mg.

How many pack sizes does BI-671800 come in?

BI-671800 is available in 2 different pack sizes.

Is BI-671800 in stock?

BI-671800 is currently made to order / not held in immediate stock. Contact us for lead time.

BI-671800

Product Specifications

CAS Number

1093108-50-9

Synonyms

AP-761, Cmpd A

SKU

C07211-5mg

Target

Prostaglandin Receptor

Applications

GPCR & G Protein

Smiles

CN (C) C1=C (C (=NC (=N1) CC2=CC=C (C=C2) NC (=O) C3=CC=C (C=C3) C (F) (F) F) N (C) C) CC (=O) O

Molecular Formula

C25H26F3N5O3

Additionnal Information

BI-671800 (AP-761, Cmpd A) is a highly specific and potent antagonist of chemoattractant receptor-homologous molecule on Th2 cells (DP2/CRTH2) with IC50 of 4.5 nM and 3.7 nM for PGD2 binding to human CRTH2 and murine CRTH2, respectively. BI-671800 is associated with a small improvement in FEV1 in symptomatic controller-naïve asthma patients, and in patients on ICS.