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Alpelisib hydrochloride

Product Specifications

CAS Number

1584128-91-5

SKU

C04959-5mg

Target

PI3K

Applications

PI3K/Akt/mTOR

Molecular Formula

C19H22F3N5O2S.ClH

Additionnal Information

Alpelisib hydrochloride is a potent and selective inhibitor of PI3Kα with an IC50 of 0.005 μM, 1.2 μM, 0.29 μM, 0.25 μM for p110α, p110β, p110δ, p110γ, respectively. It exhibits good efficacy in inhibiting the growth of PI3Ka driven tumors and can be used in cancer research.

Available Sizes

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