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YW-N-7 TFA

Product Specifications

SKU

C04940-1mg

Target

C-RET

Applications

Protein Tyrosine Kinase

Additionnal Information

YW-N-7 TFA is a PROTAC that targets the inhibition and degradation of RET with a DC50 of 88 nM. It also exhibits antitumor activity in a KIF5B-RET-driven xenograft mouse model.
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