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NF449 octasodium

Product Specifications

CAS Number

627034-85-9

SKU

C04760-1mg

Additionnal Information

NF449 octasodium is a highly potent P2X1 receptor antagonist, with IC50s of 0.28, 0.69, and 120 nM for rP2X1, rP2X1+5, P2X2+3, respectively. NF449 octasodium is a Gsα-selective G Protein antagonist. NF449 octasodium suppresses the rate of GTP[γS] binding to Gsα-s, inhibits the stimulation of adenylyl cyclase activity, and blocks the coupling of β-adrenergic receptors to Gs.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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