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LE 300

Product Specifications

CAS Number

274694-98-3

SKU

C04395-1mg

Additionnal Information

LE 300 is a potent and selective dopamine D1-like receptor antagonist with Kis of 1.9 nM and 7.5 nM in CHO cell membranes expressing human dopamine D1 and D5 receptors, respectively. LE 300 is an antagonist of the 5-HT2A receptor with a pA2 of 8.32 in a rat tail artery assay.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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