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Prinaberel

Product Specifications

CAS Number

524684-52-4

Synonyms

ERB-041

SKU

C04364-5mg

Additionnal Information

Prinaberel (ERB-041) is a potent and selective estrogen receptor (ER) β agonist with IC50s of 5.4, 3.1 and 3.7 nM for human, rat and mouse ERβ, respectively. Prinaberel displays >200-fold selectivity for ERβ over ERα. Prinaberel is a potent skin cancer chemopreventive agent that acts by dampening the WNT/β-catenin signaling pathway. Prinaberel induces ovarian cancer apoptosis.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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