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MK-5046

Product Specifications

CAS Number

1022152-70-0

SKU

C04246-1mg

Additionnal Information

MK-5046 is a potent, selective and orally active Bombesin receptor subtype-3 (BRS-3) allosteric agonist with an IC50 and an EC50 value of 27 and 25 nM for hBRS-3, respectively. MK-5046 inhibits food intake and reduces body weight of diet-induced obese (DIO) mouse models. MK-5046 can be used for the research of obesity.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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