What is the catalog number for Phentolamine hydrochloride?

The catalog number for Phentolamine hydrochloride is C03693.

What sizes are available for Phentolamine hydrochloride?

Phentolamine hydrochloride is available in the following size(s): 5 mg, 25 mg, 100 mg, 1 g.

How many pack sizes does Phentolamine hydrochloride come in?

Phentolamine hydrochloride is available in 4 different pack sizes.

Is Phentolamine hydrochloride in stock?

Phentolamine hydrochloride is currently made to order / not held in immediate stock. Contact us for lead time.

Phentolamine hydrochloride

Product Specifications

CAS Number

73-05-2

SKU

C03693-5mg

Target

Adrenergic Receptor

Applications

Neuronal Signaling

Additionnal Information

Phentolamine hydrochloride is a potent, selective, and orally active antagonist of α1 and α2 adrenergic receptors , with pKi values of 8.8, 8.0, and 8.3 for the human α2A, α2B, and α2C adrenergic receptors, respectively. It also shows binding affinities for the α1-adrenoceptor subtypes, exhibiting Ki values of 6.1 nM for cloned α1A/D, 39.8 nM for α1B, and 2.8 nM for α1C.