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CAY10499

Product Specifications

CAS Number

359714-55-9

Synonyms

MAGL-IN-5

SKU

C03568-5mg

Target

Lipase

Applications

Metabolism

Additionnal Information

CAY10499 (MAGL-IN-5) is a non-selective lipase inhibitor with IC50 values of 144 nM for human recombinant monoacylglycerol lipase (MAGL), 90 nM for hormone-sensitive lipase (HSL), and 14 nM for fatty acid amide hydrolase (FAAH) . It also inhibits cell growth in MCF-7, MB-231, COV318, OVCAR-3 cancer cell lines.
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