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Vorapaxar sulfate

Product Specifications

CAS Number

705260-08-8

Synonyms

SCH 530348 sulfate

SKU

C03395-5mg

Target

PAR

Applications

GPCR & G Protein

Additionnal Information

Vorapaxar sulfate (SCH 530348 sulfate) is a selective and orally active antagonist of protease-activated receptor (PAR-1), with a Ki value of 8.1 nM. Vorapaxar sulfate reduces thrombin receptor-activating peptide (TRAP) -induced platelet aggregation in a dose-dependent manner.

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