Tacrine
Product Specifications
CAS Number
321-64-2
SKU
C03377-5mg
Target
AChR
Applications
Neuronal Signaling
Additionnal Information
Tacrine is a potent acetylcholinesterase (AChE) inhibitor. It inhibits acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) with an IC50 of 77 nM and 69 nM, respectively. It is used in the treatment of Alzheimer's disease (AD), also poisoning topoisomerases and inhibiting in vivo (mitochondrial) mtDNA synthesis.
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