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YJ1206

Product Specifications

CAS Number

3053716-98-3

SKU

C03332-5mg

Target

CDK

Applications

Cell Cycle

Additionnal Information

YJ1206 is an orally bioavailable, highly specific and potent degrader of CDK12/13 with an IC50 of 12.55 nM in VCaP cells. It increases DNA damage, induces apoptosis, and demonstrates robust anti-tumor activity in vivo.

Available Sizes

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