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GSK-2879552

Product Specifications

CAS Number

1401966-69-5

SKU

C03216-5mg

Target

LSD1

Applications

Epigenetics

Additionnal Information

GSK-2879552 is a selective and potent inhibitor of Lysine-specific demethylase 1 (LSD1, KDM1A), with the potential to treat Small cell lung cancer (SCLC) . It induces the expression of putative KDM1A target genes and demonstrates potent, predominantly cytostatic, antiproliferative activity in SCLC cell lines and tumor xenograft models.

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