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Cabotegravir Sodium

Product Specifications

CAS Number

1051375-13-3

Synonyms

GSK-1265744 sodium

SKU

C03198-5mg

Target

Integrase

Applications

Microbiology

Additionnal Information

Cabotegravir (GSK-1265744) sodium is a orally active and long-acting HIV integrase strand transfer inhibitor. It also inhibits organic anion transporter 1/3 (OAT1/OAT3) with IC50 of 0.41 μM and 0.81 μM for OAT3 and OAT1, respectively.

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