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Cirtuvivint

Product Specifications

CAS Number

2143917-62-6

Synonyms

SM08502

SKU

C02148-5mg

Target

CDK

Applications

Cell Cycle

Additionnal Information

Cirtuvivint (SM08502) is a potent and orally active inhibitor of CDC-like kinase (CLK) and a DYRK (dual-specificity tyrosine kinase) that targets mRNA splicing and is optimized for Wnt pathway inhibition. Cirtuvivint inhibits serine and arginine-rich splicing factor (SRSF) phosphorylation and disrupts spliceosome activity. Cirtuvivint can be used for solid tumor research.

Available Sizes

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