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GNE 2861

Product Specifications

CAS Number

1394121-05-1

SKU

C02063-5mg

Target

PAK

Applications

Cytoskeletal Signaling

Smiles

COCCNC1=NC2=C (C=C (C=C2) C#CC3 (O) CCCCC3) [N]1C4=NC (=NC=C4) N

Additionnal Information

GNE 2861, a PAK inhibitor that displays group II selectivity, inhibits PAK4, PAK5 and PAK6 with IC50s of 7.5, 36, 126 nM, respectively.

Storage Conditions

3 years -20°C powder

Available Sizes

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