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KY-05009

Product Specifications

CAS Number

1228280-29-2

SKU

C02059-5mg

Target

MAP4K

Applications

MAPK

Smiles

CC1=CC=C (C=C1) C (=O) NC2=C (N=C (NC3=CC=CC=C3) S2) C (N) =O

Additionnal Information

KY-05009 is an ATP-competitive Traf2- and Nck-interacting kinase (TNIK) inhibitor with a Ki of 100 nM, which inhibits the protein expression of TNIK and transcriptional activity of Wnt target genes and induces apoptosis in cancer cells.

Storage Conditions

3 years -20°C powder

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