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BBI-355

Product Specifications

CAS Number

2871056-82-3

SKU

C02004-5mg

Target

Chk

Applications

Cell Cycle

Additionnal Information

BBI-355 is an oral, potent, and selective small molecule inhibitor of CHK1 with an IC50 of 0.3 nM. It demonstrates significant anti-tumor activity as a single agent and in combination with targeted therapies in multiple ecDNA+ oncogene amplified tumor models.

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