What is the catalog number for MS8709?

The catalog number for MS8709 is C01991.

What sizes are available for MS8709?

MS8709 is available in the following size(s): 5 mg, 25 mg, 100 mg, 1 g.

How many pack sizes does MS8709 come in?

MS8709 is available in 4 different pack sizes.

MS8709 is currently made to order / not held in immediate stock. Contact us for lead time.

MS8709

Product Specifications

CAS Number

3060730-06-2

Synonyms

EX-A11295

SKU

C01991-5mg

Target

G9a/GLP

Applications

Epigenetics

Additionnal Information

MS8709 (EX-A11295) is a first-in-class G9a/GLP proteolysis targeting chimera (PROTAC) degrader, that induces G9a/GLP degradation in a concentration, time, and ubiquitin-proteasome system (UPS) -dependent manner, and does not alter the mRNA expression of G9a/GLP over other methyltransferases. It displays superior cell growth inhibition in prostate, leukemia, and lung cancer cells over parent G9a/GLP inhibitors.