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IK-930

Product Specifications

CAS Number

2563892-44-2

SKU

C01698-5mg

Target

TEAD

Applications

Hippo

Additionnal Information

IK-930 is a selective, small-molecule inhibitor of TEAD that prevents palmitate binding and thereby disrupts aberrant TEAD-dependent transcription. IK-930 demonstrates antitumor activity in mouse xenograft models with Hippo pathway genetic alterations.

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