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Talnetant

Product Specifications

CAS Number

174636-32-9

Synonyms

SB 223412

SKU

C01670-5mg

Additionnal Information

Talnetant (SB 223412) is a selective, competitive, brain-permeable NK3 receptor antagonist with a Ki of 1.4 nM in hNK-3-CHO cells. Talnetant is 100-fold more selective for hNK-3 relative to the hNK-2 receptor and has no affinity for hNK-1. Talnetant can be used in schizophrenia-related studies.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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