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Imlunestrant

Product Specifications

CAS Number

2408840-26-4

Synonyms

LY3484356

SKU

C01603-5mg

Target

Estrogen/progestogen Receptor

Applications

Endocrinology & Hormones

Additionnal Information

Imlunestrant (LY3484356) is a potent, orally bioavailable selective estrogen receptor degrader (SERD) that functions as a pure antagonist of estrogen receptor alpha (ERα) . It inhibits ER-dependent gene transcription and cell proliferation, resulting in sustained suppression of estrogen-driven growth in ER-positive cells.

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