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CFT8634

Product Specifications

CAS Number

2704617-96-7

SKU

C01527-5mg

Target

Epigenetic Reader Domain

Applications

Epigenetics

Additionnal Information

CFT8634 is a potent BRD9 degrader with DC50 of 3 nM. It forms a ternary complex with BRD9 and an E3 ligase, resulting in BRD9 ubiquitination. CFT8634 is used in the treatment of SMARCB1-perturbed cancers.

Storage Conditions

3 years -20°C powder

Available Sizes

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