What is the catalog number for Relacorilant (CORT125134)?

The catalog number for Relacorilant (CORT125134) is C01471.

What sizes are available for Relacorilant (CORT125134)?

Relacorilant (CORT125134) is available in the following size(s): 5 mg, 10 mM / 1 mL, 25 mg, 100 mg.

How many pack sizes does Relacorilant (CORT125134) come in?

Relacorilant (CORT125134) is available in 4 different pack sizes.

Is Relacorilant (CORT125134) in stock?

Relacorilant (CORT125134) is currently made to order / not held in immediate stock. Contact us for lead time.

Relacorilant (CORT125134)

Product Specifications

CAS Number

1496510-51-0

SKU

C01471-5mg

Target

Glucocorticoid Receptor

Applications

Endocrinology & Hormones

Smiles

C[N]1C=C (C=N1) [S; v6] (=O) (=O) N2CCC3=CC4=C (CC3 (C2) C (=O) C5=CC (=CC=N5) C (F) (F) F) C=N[N]4C6=CC=C (F) C=C6

Additionnal Information

Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.