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ERG240

Product Specifications

CAS Number

1415683-79-2

SKU

C01431-5mg

Target

Transferase

Applications

Metabolism

Smiles

[Na; v0].CC (CCC (O) =O) C (C) =O

Additionnal Information

ERG240, a selective inhibitor of branched-chain aminotransferase 1 (BCAT1) with an IC50 of 0.1-1nM, leads to decreased oxygen consumption and glycolysis through the down regulation of IRG1 expression, which leads to decrease itaconate production in human macrophages.

Storage Conditions

3 years -20°C powder

Available Sizes

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