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Zapnometinib (PD0184264)

Product Specifications

CAS Number

303175-44-2

Synonyms

ATR-002

SKU

C01234-5mg

Target

MEK

Applications

Protein Tyrosine Kinase

Smiles

OC (=O) C1=C (NC2=C (Cl) C=C (I) C=C2) C (=C (F) C=C1) F

Additionnal Information

Zapnometinib (PD0184264, ATR-002), an major active metabolite of CI-1040, is a novel MEK inhibitor with an IC50 of 5.7 nM.

Storage Conditions

3 years -20°C powder

Available Sizes

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