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AS1269574

Product Specifications

CAS Number

330981-72-1

SKU

C01203-5mg

Target

GPR

Applications

GPCR & G Protein

Smiles

CC1=CC (=NC (=N1) C2=CC=C (Br) C=C2) NCCO

Additionnal Information

AS 1269574, a small-molecule G protein-coupled receptor 119 (GPR119) agonist, has an EC50 of 2.5 μM in HEK293 cells transiently expressing human GPR119 and enhances insulin secretion in the mouse pancreatic β-cell line MIN-6 only under high-glucose (16.8 mM) conditions.

Storage Conditions

3 years -20°C powder

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