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Ivarmacitinib

Product Specifications

CAS Number

1445987-21-2

Synonyms

SHR0302

SKU

C01188-5mg

Target

JAK

Applications

Angiogenesis

Additionnal Information

Ivarmacitinib (SHR0302) is a potent and orally active inhibitor of JAK family, particularly JAK1. Ivarmacitinib demonstrates more than 10-fold selectivity for JAK1 over JAK2, 77-fold over JAK3, and 420-fold over Tyk2. Ivarmacitinib also exhibits anti-proliferative and anti-inflammatory effects.

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