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ML401

Product Specifications

CAS Number

1597489-14-9

SKU

C01071-5mg

Target

GPR

Applications

GPCR & G Protein

Smiles

ClC1=CC=C (CN2CCN (CC2) C (=O) \C=C\C3=CC=C (Br) C=C3) C=C1

Additionnal Information

ML401, a potent chemical probe, selectively antagonizes G-protein coupled receptor 183 (GPR183, EBI2) with an IC50 of 1.03 nM, and displays activity in a chemotaxis assay with IC50 of 6.24 nM.

Storage Conditions

3 years -20°C powder

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