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ICA-27243

Product Specifications

CAS Number

325457-89-4

SKU

C01070-5mg

Target

Potassium Channel

Applications

Transmembrane Transporters

Smiles

FC1=C (F) C=C (C=C1) C (=O) NC2=CN=C (Cl) C=C2

Additionnal Information

ICA-27243, a selective activator of the neuronal M current and KCNQ2/Q3 channels, induces a concentration-dependent increase in a 86Rb+ efflux from CHO cells expressing KCNQ2/Q3 channels with EC50 of 0.2 μM.

Storage Conditions

3 years -20°C powder

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