SR 16584

SR 16584 is a selective antagonist of α3β4 nAChR with an IC50 of 10.2 μM[1].

Product Specifications

CAS Number

[1150153-86-8]

UNSPSC

12352005

Target

NAChR

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/sr-16584.html

Solubility

10 mM in DMSO

Smiles

O=C1N([C@@H]2C[C@@H]3N(C)[C@@H](CCC3)C2)C4=CC=CC=C4C1

Molecular Formula

C17H22N2O

Molecular Weight

270.37

References & Citations

[1]Zaveri N, et al. Novel α3β4 nicotinic acetylcholine receptor-selective ligands. Discovery, structure-activity studies, and pharmacological evaluation. J Med Chem. 2010 Nov 25;53 (22) :8187-91.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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