Protegrin-1
Protegrin-1 is an orally active antibacterial peptide. Protegrin-1 activates ERK, COX2, NFκB, inhibits Apoptosis, and NO production. Protegrin-1 has antibacterial activity against S. aureus, E. faecium, E. coli, P. aeruginosa and K. Pneumoniae, with MBC values between 10 and 20 µM. Protegrin-1 has antiviral activity against dengue NS2B-NS3. Protegrin-1 has anti-inflammatory activity. Protegrin-1 is used in the study of inflammatory diseases and infections[1][2][3][4][5][6][7][8].
Product Specifications
CAS Number
168831-77-4
Product Name Alternative
PG1
UNSPSC
12352209
Target
Apoptosis; Bacterial; COX; Dengue Virus; ERK; NF-κB; NO Synthase
Type
Peptides
Related Pathways
Anti-infection; Apoptosis; Immunology/Inflammation; MAPK/ERK Pathway; NF-κB; Stem Cell/Wnt
Field of Research
Infection; Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/protegrin-1.html
Purity
99.55
Solubility
DMSO : 20 mg/mL (ultrasonic)
Smiles
Molecular Formula
C88H147N37O19S4
Molecular Weight
2155.61
References & Citations
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Scientific Category
Peptides
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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