Vapreotide
Vapreotide is a neurokinin-1 (NK1) receptor antagonist, with an IC50 of 330 nM.
Product Specifications
CAS Number
[103222-11-3]
Product Name Alternative
RC160; BMY 41606
UNSPSC
12352209
Target
Neurokinin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/Vapreotide.html
Purity
99.87
Solubility
H2O : ≥ 100 mg/mL
Smiles
O=C([C@@H](NC([C@H](CSSC[C@H](NC([C@@H](NC([C@@H](NC1=O)CCCCN)=O)C(C)C)=O)C(N[C@H](C(N)=O)CC2=CNC3=CC=CC=C23)=O)NC([C@H](N)CC4=CC=CC=C4)=O)=O)CC5=CC=C(C=C5)O)N[C@@H]1CC6=CNC7=CC=CC=C67
Molecular Formula
C57H70N12O9S2
Molecular Weight
1131.37
References & Citations
[1]Spitsin S et al. Analog of somatostatin vapreotide exhibits biological effects in vitro via interaction with neurokinin-1 receptor. Neuroimmunomodulation. 2013;20 (5) :247-55.
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture and light)
Scientific Category
Peptides
Clinical Information
Launched
Isoform
NK1R
Available Sizes
Curated Selection
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