Umbralisib R-enantiomer
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is a PI3Kδ inhibitor, which is the less active enantiomer of TGR-1202.
Product Specifications
CAS Number
[1532533-69-9]
Product Name Alternative
TGR-1202 R-enantiomer; RP5264 R-enantiomer
UNSPSC
12352005
Target
PI3K
Type
Reference compound
Related Pathways
PI3K/Akt/mTOR
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/TGR-1202-R-enantiomer.html
Concentration
10mM
Purity
99.52
Solubility
DMSO : 33.33 mg/mL (ultrasonic)
Smiles
O=C1C(C2=CC=CC(F)=C2)=C([C@@H](C)N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)OC6=CC=C(F)C=C16
Molecular Formula
C31H24F3N5O3
Molecular Weight
571.55
References & Citations
[1]Michael Weiss, et al. Combination of anti-cd20 antibody and pi3 kinase selective inhibitor. WO2014071125A1.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
PI3Kδ
Available Sizes
Curated Selection
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