PKM2-IN-5
PKM2-IN-5 (Compound G1) is an inhibitor for pyruvate kinase M2 (PKM2), with IC50 >70 μM[1].
Product Specifications
CAS Number
904457-46-1
UNSPSC
12352005
Target
Pyruvate Kinase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/pkm2-in-5.html
Solubility
10 mM in DMSO
Smiles
O=C1OC2=C(C3=C1C=C(C(NC(C)C)=O)S3)C=C(C)C=C2
Molecular Formula
C16H15NO3S
Molecular Weight
301.36
References & Citations
[1]Cantley L, et al., Inhibitors of pyruvate kinase and methods of treating disease. WO2008019139
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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