PKM2-IN-5
PKM2-IN-5 (Compound G1) is an inhibitor for pyruvate kinase M2 (PKM2), with IC50 >70 μM[1].
Product Specifications
CAS Number
904457-46-1
UNSPSC
12352005
Target
Pyruvate Kinase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/pkm2-in-5.html
Solubility
10 mM in DMSO
Smiles
O=C1OC2=C(C3=C1C=C(C(NC(C)C)=O)S3)C=C(C)C=C2
Molecular Formula
C16H15NO3S
Molecular Weight
301.36
References & Citations
[1]Cantley L, et al., Inhibitors of pyruvate kinase and methods of treating disease. WO2008019139
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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