LY206130 (free base)
LY206130 free base is a 5-HT1A receptor antagonist with the activity of enhancing exogenous serotonin levels. LY206130 free base, when used concomitantly with fluoxetine, may enhance the appetite-suppressing effects of fluoxetine. LY206130 free base was shown to significantly reduce sweetened milk concentrate consumption in a dietary model. Clinical application of LY206130 free base may be beneficial in curbing eating disorders and obesity[1].
Product Specifications
CAS Number
127414-58-8
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ly206130-free-base.html
Smiles
OC(CNC1CCCCC1)COC2=CC=CC3=C2C=CN3
Molecular Formula
C17H24N2O2
Molecular Weight
288.38
References & Citations
[1]5HT1A receptor antagonists enhance the functional activity of fluoxetine in a mouse model of feeding
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT1 Receptor
Frequently Asked Questions
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