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CDK8-IN-14

CDK8-IN-14 (compound 12) inhibits CDK8 with an IC50 value of 39.2 nM and has anti-AML cell proliferation activity (molm-13 GC50 = 0.02±0.01μM, MV4-11 GC50 = 0.03±0.01μM) [1].

Product Specifications

CAS Number

[2924193-12-2]

UNSPSC

12352005

Target

CDK

Type

Reference compound

Related Pathways

Cell Cycle/DNA Damage

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/cdk8-in-14.html

Solubility

10 mM in DMSO

Smiles

O=C(N)C1=CC=CC(C2=CN=C(NC=C3C4=COC=C4)C3=C2)=C1

Molecular Formula

C18H13N3O2

Molecular Weight

303.31

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Curated Selection

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