Fotagliptin (benzoate)
Fotagliptin benzoate is a Dipeptidyl Peptidase IV (DPP-4) inhibitor (IC50=2.27 nM) . Fotagliptin benzoate displays great security in rat and dog. Fotagliptin benzoate can be used for Type 2 diabetes mellitus research[1].
Product Specifications
CAS Number
[1403496-40-1]
Product Name Alternative
SAL067
UNSPSC
12352005
Target
Dipeptidyl Peptidase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/fotagliptin-benzoate.html
Purity
99.19
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
OC(C1=CC=CC=C1)=O.CC(C2=O)=NN=C(N3C[C@@H](CCC3)N)N2CC4=C(C=CC(F)=C4)C#N
Molecular Formula
C24H25FN6O3
Molecular Weight
464.49
References & Citations
[1]Wang Z, et al. Development and validation of a UPLC-MS/MS method for simultaneous determination of fotagliptin and its two major metabolites in human plasma and urine. Bioanalysis. 2017 Feb;9 (4) :381-393.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture and light)
Scientific Category
Reference compound1
Clinical Information
Phase 3
Isoform
DPP-4
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
043284-ML750 100 µL
TRPC1, CT (TRPC1, TRP1, Short transient receptor potential channel 1, Transient receptor protein 1) (MaxLight 750) discontinued
Ask
View Details QP9948-iv-50ug 50ug
Recombinant Human Beta-2 adrenergic receptor Protein, His-SUMO, Invitro-E.coli-50ug
Ask
View Details DML20-1000ML 1000 mL
DMEM (HG) With high-glucose. W/O L-glutamine, sodium pyruvate and phenol red.
Ask
View Details 
KTE61783-01 48 Tests
Human Low-density lipoprotein receptor-related protein 2 (LRP2) ELISA Kit
Ask
View Details KTE61783-02 96 Tests
Human Low-density lipoprotein receptor-related protein 2 (LRP2) ELISA Kit
Ask
View Details