CB1 agonist 1

CB1 agonist 1 (compound 22) is an agonist of CB1. CB1 agonist 1 shows affinity to CB1 receptor with an pIC50 value of 5.7. CB1 agonist 1 can be used for the research of brain disorders[1].

Product Specifications

CAS Number

[851212-80-1]

UNSPSC

12352005

Hazard Statement

H302, H315, H319

Target

Cannabinoid Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/cb1-agonist-1.html

Purity

99.84

Solubility

DMSO : 250 mg/mL (ultrasonic)

Smiles

O=C(C1=C(OC2=CC=CC=C2)C=CC=C1)NC3=CC=C(C)C(S(=O)(N4CCOCC4)=O)=C3

Molecular Formula

C24H24N2O5S

Molecular Weight

452.52

Precautions

H302, H315, H319

References & Citations

[1]Lambeng N, et al. Arylsulfonamides as a new class of cannabinoid CB1 receptor ligands: identification of a lead and initial SAR studies. Bioorg Med Chem Lett. 2007 Jan 1;17 (1) :272-7.