(d (CH2) 51, Tyr (Me) 2, Dab5, Arg8) -Vasopressin
(d (CH2) 51, Tyr (Me) 2, Dab5, Arg8) -Vasopressin (d (CH2) 5[Tyr (Me) 2, Dab5]AVP) is a specific antagonist of vasopressin V1a receptor, with a pA2 of 6.71[1].
Product Specifications
CAS Number
176714-12-8
Product Name Alternative
D (CH2) 5[Tyr (Me) 2, Dab5]AVP
UNSPSC
12352209
Target
Vasopressin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/d-ch2-51-tyr-me-2-dab5-arg8-vasopressin.html
Solubility
10 mM in DMSO
Smiles
O=C1CC2(CCCCC2)SSC[C@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](N1)CC3=CC=C(C=C3)OC)=O)CC4=CC=CC=C4)=O)CCC(N)=O)=O)CCN)=O)C(N5[C@@H](CCC5)C(N[C@H](C(NCC(N)=O)=O)CCCNC(N)=N)=O)=O
Molecular Formula
C52H76N14O11S2
Molecular Weight
1137.38
References & Citations
[1]Chan WY, et, al. Discovery and design of novel and selective vasopressin and oxytocin agonists and antagonists: the role of bioassays. Exp Physiol. 2000 Mar;85 Spec No:7S-18S.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
BNC470965-100 1x 100 µL
MUC1 / CA15-3 / EMA / CD227 (Epithelial Marker) (VU-11D1), CF647 conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC400204-100 1x 100 µL
Complement C4d (C4D204), CF640R conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC941386-500 1x 500 µL
Ferritin, Light Chain (FTL) (Microglia Marker) (FTL/1386), CF594 conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
BNC940714-500 1x 500 µL
Thymidylate Synthase (TS106), CF594 conjugate, 0.1mg/mL
Sign In for Pricing
View Details