(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
Product Specifications
UNSPSC Description
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin (d(CH2)5[Tyr(Me)2, Dab5]AVP) is a specific antagonist of vasopressin V1a receptor, with a pA2 of 6.71[1].
Target Antigen
Vasopressin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/d-ch2-51-tyr-me-2-dab5-arg8-vasopressin.html
Solubility
10 mM in DMSO
Smiles
O=C1CC2(CCCCC2)SSC[C@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](N1)CC3=CC=C(C=C3)OC)=O)CC4=CC=CC=C4)=O)CCC(N)=O)=O)CCN)=O)C(N5[C@@H](CCC5)C(N[C@H](C(NCC(N)=O)=O)CCCNC(N)=N)=O)=O
Molecular Weight
1137.38
References & Citations
[1]Chan WY, et, al. Discovery and design of novel and selective vasopressin and oxytocin agonists and antagonists: the role of bioassays. Exp Physiol. 2000 Mar;85 Spec No:7S-18S.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-P5006/d-CH2-51-Tyr-Me-2-Dab5-Arg8-Vasopressin-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-P5006/
Clinical Information
No Development Reported
CAS Number
176714-12-8
Curated Selection
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