KSCM-1
Product Specifications
UNSPSC Description
KSCM-1 is a selective sigma-1 receptor ligand with a Ki of 27.5 nM. KSCM-1 shows more selective for sigma-1 over sigma-2, and shows no significant affinity at non-sigma receptors[1].
Target Antigen
Sigma Receptor
Type
Reference compound
Related Pathways
Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/kscm-1.html
Smiles
O=C(N(CCCN1CCCCC1)C2=CC=CC=C2)C3=C(C4=CC(OC)=C(C=C4O3)OC)C
Molecular Weight
436.54
References & Citations
[1]Karla-Sue C Marriott, et al. Synthesis of N-phenyl-N-(3-(piperidin-1-yl)propyl)benzofuran-2-carboxamides as new selective ligands for sigma receptors. Bioorg Med Chem. 2012 Dec 1;20(23):6856-61.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-118279/KSCM-1-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-118279/
Clinical Information
Phase 1
CAS Number
1415247-17-4
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items