Methapyrilene (fumarate)

Methapyrilene fumarate is a histamine receptor H1 antagonist. Methapyrilene fumarate has sedative effects. Methapyrilene fumarate is being studied for its analgesic properties[1].

Product Specifications

CAS Number

[33032-12-1]

UNSPSC

12352005

Target

Histamine Receptor

Related Pathways

GPCR/G Protein; Immunology/Inflammation; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Smiles

CN(C)CCN(C1=CC=CC=N1)CC2=CC=CS2.OC(/C=C/C(O)=O)=O.[1.5]

Molecular Formula

C20H25N3O6S

Molecular Weight

435.50

References & Citations

[1]Smith GM, et al. Use of subjective responses to evaluate efficacy of mild analgesic-sedative combinations. Clin Pharmacol Ther. 1974 Feb;15 (2) :118-29.